Granules India Limited has high volume world-class facilities for APIs, PFIs, & FDFs, serving customers in over 80 countries.

Contact Supplier

Jai Radhe Sales is your partner for all your sourcing needs.

ACCESS ALL DATA
Browse all information
CHEMISTRY
Discover Molecule Insights

ACTIVE PHARMA INGREDIENTS

1 API Suppliers, 1 Listed Suppliers, $ API Reference Price

1 API Suppliers
1 Listed Suppliers
$ API Reference Price

DIGITAL CONTENT

3 NEWS #PharmaBuzz

media
3 NEWS #PharmaBuzz

Synopsis

ACTIVE PHARMA INGREDIENTS

API Suppliers

USDMF

CEP/COS

JDMF

EU WC

KDMF

NDC API

VMF

Listed Suppliers

API REF. PRICE (USD/KG)

$ 5,278

MARKET PLACE

API

FDF

0INTERMEDIATES

FINISHED DOSAGE FORMULATIONS

FDF Dossiers

FDA Orange Book

Europe

Canada

Australia

South Africa

Listed Dossiers

0 DRUGS IN DEVELOPMENT

DRUG PRODUCT COMPOSITIONS

REF. STANDARDS OR IMPURITIES

EDQM

USP

Others

PATENTS & EXCLUSIVITIES

US Patents

US Exclusivities

Health Canada Patents

DIGITAL CONTENT

Data Compilation #PharmaFlow

Stock Recap #PipelineProspector

Weekly News Recap #Phispers

News #PharmaBuzz

GLOBAL SALES INFORMATION

US Medicaid (USD)

Annual Reports (USD Million)

Finished Drug Prices

0RELATED EXCIPIENT COMPANIES

0EXCIPIENTS BY APPLICATIONS

Chemistry

Click the arrow to open the dropdown

Click the button for full data set

Also known as: 1165910-22-4, Lgd-4033, Ligandrol, Lgd4033, Vk-5211, 4-[(2r)-2-[(1r)-2,2,2-trifluoro-1-hydroxyethyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile

Molecular Formula

C₁₄H₁₂F₆N₂O

Molecular Weight

338.25 g/mol

InChI Key

OPSIVAKKLQRWKC-VXGBXAGGSA-N

FDA UNII

1EJT54415A

Ligandrol is an investigational selective androgen receptor modulator (SARM) for treatment of conditions such as muscle wasting and osteoporosis.

1 2D Structure

Ligandrol

2 Identification

2.1 Computed Descriptors

2.1.1 IUPAC Name

4-[(2R)-2-[(1R)-2,2,2-trifluoro-1-hydroxyethyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile

2.1.2 InChI

InChI=1S/C14H12F6N2O/c15-13(16,17)10-6-9(4-3-8(10)7-21)22-5-1-2-11(22)12(23)14(18,19)20/h3-4,6,11-12,23H,1-2,5H2/t11-,12-/m1/s1

2.1.3 InChI Key

OPSIVAKKLQRWKC-VXGBXAGGSA-N

2.1.4 Canonical SMILES

C1CC(N(C1)C2=CC(=C(C=C2)C#N)C(F)(F)F)C(C(F)(F)F)O

2.1.5 Isomeric SMILES

C1C[C@@H](N(C1)C2=CC(=C(C=C2)C#N)C(F)(F)F)[C@H](C(F)(F)F)O

2.2 Other Identifiers

2.2.1 UNII

1EJT54415A

2.3 Synonyms

2.3.1 MeSH Synonyms

1. 4-(2-(2,2,2-trifluoro-1-hydroxyethyl)pyrrolidin-1-yl)-2-(trifluoromethyl)benzonitrile

2. Lgd-4033

2.3.2 Depositor-Supplied Synonyms

1. 1165910-22-4

2. Lgd-4033

3. Ligandrol

4. Lgd4033

5. Vk-5211

6. 4-[(2r)-2-[(1r)-2,2,2-trifluoro-1-hydroxyethyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile

7. 1ejt54415a

8. 4-[(2r)-2-[(1r)-2,2,2-trifluoro-1-hydroxyethyl]-1-pyrrolidinyl]-2-(trifluoromethyl)benzonitrile

9. Unii-1ejt54415a

10. 4-((2r)-2-((1r)-2,2,2-trifluoro-1-hydroxyethyl)-1-pyrrolidinyl)-2-(trifluoromethyl)benzonitrile

11. 4-{(2r)-2-[(1r)-2,2,2-trifluoro-1-hydroxyethyl]-1-pyrrolidinyl}-2-(trifluoromethyl)benzonitrile

12. Benzonitrile, 4-((2r)-2-((1r)-2,2,2-trifluoro-1-hydroxyethyl)-1-pyrrolidinyl)-2-(trifluoromethyl)-

13. Benzonitrile, 4-[(2r)-2-[(1r)-2,2,2-trifluoro-1-hydroxyethyl]-1-pyrrolidinyl]-2-(trifluoromethyl)-

14. Ligandrol;lgd-4033

15. Schembl221159

16. Ligandrol [nflis-drug]

17. Lgd4033(lg)

18. Vk5211

19. Dtxsid10657620

20. Ex-a729

21. Bcp07128

22. Lgd-4033lgd-4033

23. Mfcd27923016

24. S8822

25. Zinc95830588

26. Akos022173564

27. Cs-4667

28. Db13934

29. Lgd-4033(vk-5211)

30. Ac-30218

31. Hy-13981

32. A14346

33. J-690039

34. Q21098841

2.4 Create Date

2009-08-10

3 Chemical and Physical Properties

Molecular Formula	C₁₄H₁₂F₆N₂O
Molecular Weight	338.25 g/mol
XLogP3	3.7
Hydrogen Bond Donor Count	1
Hydrogen Bond Acceptor Count	9
Rotatable Bond Count	2
Exact Mass	338.08538198 g/mol
Monoisotopic Mass	338.08538198 g/mol
Topological Polar Surface Area	47.3 Å²
Heavy Atom Count	23
Formal Charge	0
Complexity	468
Isotope Atom Count	0
Defined Atom Stereocenter Count	2
Undefined Atom Stereocenter Count	0
Defined Bond Stereocenter Count	0
Undefined Bond Stereocenter Count	0
Covalently Bonded Unit Count	1

API SUPPLIERS

FULL SCREEN VIEW Click here to open all results in a new tab [this preview display 10 results]

Listed Suppliers

FULL SCREEN VIEW Click here to open all results in a new tab [this preview display 10 results]

API Reference Price

[{"dataSource":"API Import","activeIngredients":"LIGANDROL","year":"2021","qtr":"Q2","strtotime":1621881000,"product":"LIGANDROL (LGD4033)","address":"12\/12, SHAKTI NAGAR,","city":"DELHI","supplier":"GREENBELT INTERNATIONAL CO. ","supplierCountry":"CHINA","foreign_port":"HONG KONG","customer":"COOPER LAB","customerCountry":"INDIA","quantity":"1.00","actualQuantity":"1","unit":"KGS","unitRateFc":"5870","totalValueFC":"5938.2","currency":"USD","unitRateINR":"434967","date":"25-May-2021","totalValueINR":"434967","totalValueInUsd":"5938.2","indian_port":"DELHI AIR","hs_no":"29371900","bill_no":"4080601","productDescription":"API","marketType":"REGULATED MARKET","country":"CHINA","selfForZScoreResived":"Pharma Grade","supplierPort":"HONG KONG","supplierAddress":"","customerAddress":"12\/12, SHAKTI NAGAR,"},{"dataSource":"API Import","activeIngredients":"","year":"2024","qtr":"Q1","strtotime":1705861800,"product":"LIGANDROL LGD-4033","address":"12\/12, SHAKTI NAGAR,","city":"DELHI","supplier":"WAHSUN PHARMACEUTICAL CO., LTD","supplierCountry":"CHINA","foreign_port":"HONG KONG","customer":"COOPER LAB","customerCountry":"INDIA","quantity":"0.55","actualQuantity":"0.55","unit":"KGS","unitRateFc":"4780","totalValueFC":"2660.3","currency":"USD","unitRateINR":"401998","date":"22-Jan-2024","totalValueINR":"221098.9","totalValueInUsd":"2660.3","indian_port":"Delhi Air","hs_no":"29371900","bill_no":"9778915","productDescription":"API","marketType":"REGULATED MARKET","country":"CHINA","selfForZScoreResived":"Pharma Grade","supplierPort":"HONG KONG","supplierAddress":"2 ND FLOOR, NO. 1830, HUQING ROAD,QINGPU DISTRICT, SHANGHAISDNF CN","customerAddress":"12\/12, SHAKTI NAGAR,"},{"dataSource":"API Import","activeIngredients":"","year":"2024","qtr":"Q4","strtotime":1729794600,"product":"LIGANDROL (LGD 4033)","address":"12\/12, SHAKTI NAGAR,","city":"DELHI","supplier":"WAHSUN PHARMACEUTICAL CO., LTD","supplierCountry":"CHINA","foreign_port":"HONG KONG","customer":"COOPER LAB","customerCountry":"INDIA","quantity":"0.61","actualQuantity":"0.612","unit":"KGS","unitRateFc":"4600","totalValueFC":"2846.1","currency":"USD","unitRateINR":"390770","date":"25-Oct-2024","totalValueINR":"239151.24","totalValueInUsd":"2846.1","indian_port":"Delhi Air","hs_no":"29371900","bill_no":"6337044","productDescription":"API","marketType":"REGULATED MARKET","country":"CHINA","selfForZScoreResived":"Pharma Grade","supplierPort":"HONG KONG","supplierAddress":"2 ND FLOOR, NO. 1830, HUQING ROAD, QINGPU DISTRICT, SHANGHAI SDNF CN","customerAddress":"12\/12, SHAKTI NAGAR,"}]

Number of Transactions

Total Quantity (KGS)

Total Value (USD)

Quantity (KGS) & Unit rate (USD/KGS) over time

API Imports and Exports

Importing Country	Total Quantity (KGS)	Average Price (USD/KGS)	Number of Transactions

Upgrade, download data, analyse, strategize, subscribe with us contact

Digital Content

Create Content with PharmaCompass, ask us

NEWS #PharmaBuzz

ABOUT THIS PAGE

Find Ligandrol manufacturers, exporters & distributors on PharmaCompass

Ligandrol

ACCESS ALL DATA

Browse all information

CHEMISTRY

Discover Molecule Insights

ACTIVE PHARMA INGREDIENTS

1 API Suppliers

1 Listed Suppliers

$ API Reference Price

DIGITAL CONTENT

3 NEWS #PharmaBuzz

ACTIVE PHARMA INGREDIENTS

API REF. PRICE (USD/KG)

$ 5,278

MARKET PLACE

0INTERMEDIATES

FINISHED DOSAGE FORMULATIONS

0 DRUGS IN DEVELOPMENT

DRUG PRODUCT COMPOSITIONS

REF. STANDARDS OR IMPURITIES

PATENTS & EXCLUSIVITIES

DIGITAL CONTENT

GLOBAL SALES INFORMATION

0RELATED EXCIPIENT COMPANIES

0EXCIPIENTS BY APPLICATIONS

Average Price (USD/KGS)

Number of Transactions

Total Quantity (KGS)

Total Value (USD)

Quantity (KGS) & Unit rate (USD/KGS) over time

What are you looking for?