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AZD5153 is a selective BRD4 inhibitor with a novel bivalent binding mode that inhibits both protein bromodomains, resulting in improved potency.
Lead Product(s): Momelotinib,AZD5153
Therapeutic Area: Oncology Product Name: GS-0387
Highest Development Status: Preclinical Product Type: Small molecule
Partner/Sponsor/Collaborator: GSK
Deal Size: Undisclosed Upfront Cash: Undisclosed
Deal Type: Licensing Agreement August 05, 2021